Zusammenfassung der Ressource
Neurotransmitter
- Acetycholine AcH (PRE & PARA POST)
- Norephephine NE (SYM POST)
- eprinephine
- Pre-ganlionic axons
- Synapse @ 1st sym
- --> ^or v paravert ganglion
- continue to prevertebral
- Extend or terminate @ adrenal medulla
- Adrenoceptors
- α (1,2)
- Blood Vessel
- Heart
- Thrombocytes
- Bronchi
- Kidney
- Adipocytes
- Inhibit lipolysis
- Lipolysis (triglycerides--> 3 fatty acid + glycerol
- Vasoconstriction
- Renin release (X tubular Na reabsorb)
- Dilation
- Aggregation
- ^ contractibility
- Constriction
- Dilation
- β (1,2,3)
- Sympathomimetics
Anmerkungen:
- mimic norepinephine and epinphrine
- direct on a &β
- indirectly on pre-syn terminal
- Agonist
- X selective Adrenaline
- B P +
- Bronchi Dil
- Vasopressor
Anmerkungen:
- Anaphlatic shock treatment
Anmerkungen:
- a type of allergy, cause death
- α selective
- 1- nasal decongestant
- Phenylephrine
- Ephedrine
- 2 hypotensive drugs
- clonide
- methyldopa
- β 2
- Salbutamol
Anmerkungen:
- Dilate bronchial smooth muscle
used as aerosol for Asthma
if not selective, +heart side effect
- Antagonist
- β1
- Propanolol
Anmerkungen:
- Side effect: Bronchial constriction
CardioVascular app: H. fail,
Stage fright
Hypertension
Angina
Cardiac arhythmias
- Atenolol
- Cholinomimetics
- on recpetor
- Muscarinic
- Pilocarpine
Anmerkungen:
- Eye drop
intraocular pressure -
for glaucoma 青光眼
- Amanita Muscaria 菇
Anmerkungen:
- BP v
口水 淚水 汗+
adominal pain, nausea
death due to H & lung failure