Endocrinology pharmacology

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Flashcards on Endocrinology pharmacology, created by ranranha on 19/08/2015.
ranranha
Flashcards by ranranha, updated more than 1 year ago
ranranha
Created by ranranha over 8 years ago
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Question Answer
Leuprolide GnRH analog גורם לשחרור מתמשך של GnRH בשימוש להורדת רמות טסטוסטרון וDHT "start up flare"
Finasteride 5- Alpha reductase inhibitore Treatment of BPH הורדת רמות DHT בלבד
Liraglunide GLP-1 receptor agonist Gs mediated Insulin secretion
Exenatide GLP-1 receptor agonist Gs mediated Insulin secretion
Aromatase inhibitors Anastrozole, Letrozole, Exemestane For treatment of breast cancer
NO containing Bisphosphonate Aledronate, Risedronate, Zoledronic acid
Aledronate mecchanisem FPP synthease inhibitor- osteoclast bone resorption inhibitors
Teriparotide PTH analoge
Denosumab Anti RANKL- Pre-osteoclast maturation inhibitor
Pioglitazone Rosiglitazone Thiazolidinedions
Thiazolidinedions- Mechanisem Binds to PPAR-gamma nuclear transtription regulatore. מורידים התנגדות לאינסולין בעיקר בעזרת העלאת adiponectin
Thiazolidinedions- side effects Weight gain, edema, hepatotoxicity, HF, incrise risk of fructures
Acrbose Miglitol Alpha- glucosidase inhibitors
Bromocriptine Cabergoline Dopamine agonist
Pegvisomant GH hormone receptor antagonist
Tesamorelin GHRH analog- used to treat HIV- associated lopodystrophy
Aspart, Glulisine, lispro Insulin- short acting
Detemir, Glargin Insulin- long acting
Chlorpropamide Tolbutamide First generation Sulonylureas
Glimepiride Glipizide Glyburide Second generation Sulonylureas
Sitagliptin Saxagliptin Linagliptin DDP-4 inhibitors 2 DM
Pramlintide Amylin analog- reduce gastic emptying and glucagone secretion
Canagliflozin SGLT-2 inhibitor Block reabsorbtion of glucose in PCT
Conivaptan Tolvaptan ADH antagonist- SIADH, block action of ADH at V2 recetpors
Desmopressin acetate Central diabetis insipidos
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