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BMS03-1023 Pharmacology of Cholinergic Transmissions

Evian Chai BMS03 - Nerve Signalling Inglés 17 fichas

Fichas del conjunto (17)

  1. 1How does Hemicholiniums block cholinergic transmission?Blocks the synthesis of ACh
  2. 2How does AH5283 block cholinergic transmission?Prevents storage of ACh
  3. 3Cholinergic neurotransmission uses what neurotransmitter?Acetylcholine
  4. 4How does botox block cholinergic neurotransmission?Blocks exocytosis of ACh
  5. 5What type of receptors are nicotinic receptors?Non selective cation channels
  6. 6What are the two types of nicotinic drugs?1. Skeletal muscle relaxants (antagonist)
    2. Ganglion blockers (antagonist, lower BP)
  7. 7Are skeletal muscle relaxants agonists or antagonists? Reversible or Irreversible? Competitive or Non-competitive?They are reversible competitive antagonists
  8. 8What do muscarinic agonists do?Mimic the PNS
  9. 9Which drug treats glaucoma by increasing aqueous humour flow? What kind of drug is this?Pilocarpine
    Muscarinic agonist
  10. 10What drug is a stimulant laxative? What kind of drug is this?Bethanacol
    Muscarinic agonist
  11. 11What do muscarinic antagonists do? What are their effects on the pupils?Inhibit the PNS
    Pupil dilation
  12. 12What drug is used to treat sinus bradycardia? What type of drug is this?Atropine
    Muscarinic antagonist
  13. 13Both muscarinic antagonists and B2 agonists can treat what?Asthma, as they block PNS/increase SNS effects eg. bronchodilation
  14. 14What do Inhibitors of Acetylcholinesterase do? What does it do for the PNS?Prevent the breakdown of acetylcholine to increase neurotransmission
    Increases PNS activity eg. secretions, SM tone, hypotension, bradycardia
  15. 15Which drug reverses skeletal muscle relaxants? What type of drug is this?Neostigmine
    AChE inhibitor
  16. 16What inhibitor of AchE aids Alzheimers?Donepezil
  17. 17What are the 5 main types of drugs impacting cholinergic transmission?1. Skeletal muscle relaxants (cholinergic)
    2. Ganglion blockers (cholinergic)
    3. Muscarinic agonists
    4. Muscarinic antagonists
    5. Inhibitors of AchE

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BMS03 - Nerve Signalling Fichas sobre BMS03-1023 Pharmacology of Cholinergic Transmissions, creado por Evian Chai el 22/04/2020.
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Evian Chai
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